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Benzimidazole Analogs as Potent Hypoxia Inducible Factor Inhibitors: Synthesis, Biological Evaluation, and Profiling Drug-like Properties
AIM: To develop potent HIF-1α inhibitors for potential treatment of cancer. MATERIALS AND METHODS: Chemical synthesis, HIF-luciferase assay, cytotoxic assay, platelet aggregation assay, western blot analysis, quantitative real-time PCR, aqueous solubility, protein binding, metabolic stability, and m...
Kaydedildi:
| Yayımlandı: | Anticancer Res |
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| Asıl Yazarlar: | , , , , , , , |
| Materyal Türü: | Artigo |
| Dil: | Inglês |
| Baskı/Yayın Bilgisi: |
2014
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| Konular: | |
| Online Erişim: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5346463/ https://ncbi.nlm.nih.gov/pubmed/25075010 |
| Etiketler: |
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