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When Is It Important to Measure Unbound Drug in Evaluating Nanomedicine Pharmacokinetics?

Nanoformulations have become important tools for modifying drug disposition, be it from the perspective of enabling prolonged drug release, protecting the drug molecule from metabolism, or achieving targeted delivery. When examining the in vivo pharmacokinetic properties of these formulations, most...

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Dettagli Bibliografici
Pubblicato in:Drug Metab Dispos
Autori principali: Stern, Stephan T., Martinez, Marilyn N., Stevens, David M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5118636/
https://ncbi.nlm.nih.gov/pubmed/27670412
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.073148
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