A carregar...

Roles of Residues F206 and V367 in Human CYP2B6: Effects of Mutations on Androgen Hydroxylation, Mechanism-Based Inactivation, and Reversible Inhibition

The crystal structures of human CYP2B6 indicate that Phe206 and Val367 are in close proximity to the substrate binding site and suggest that both residues may play important roles in substrate metabolism and inhibitor binding. To test this hypothesis, we investigated the effects of mutating these re...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Drug Metab Dispos
Main Authors: Lin, Hsia-lien, Zhang, Haoming, Kenaan, Cesar, Hollenberg, Paul F.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5074475/
https://ncbi.nlm.nih.gov/pubmed/27538916
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.071662
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!