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Cyclic-ketoximes as ER beta-selective agonists

The development of selective ERβ-agonists represents a therapeutic strategy against several kinds of cancers, but the high homology between the two receptor subtypes, ERα and ERβ, makes the achievement of this goal very challenging. In the past, we developed salicylaldoxime- and salicylketoxime-base...

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Библиографические подробности
Опубликовано в: :ChemMedChem
Главные авторы: Granchi, Carlotta, Lapillo, Margherita, Spena, Concetta Russo, Rizzolio, Flavio, Tuccinardi, Tiziano, Martin, Teresa A., Carlson, Kathryn E., Katzenellenbogen, John A., Minutolo, Filippo
Формат: Artigo
Язык:Inglês
Опубликовано: 2016
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4993649/
https://ncbi.nlm.nih.gov/pubmed/27135651
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201600140
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