The Philip S. Protoghese Medicinal Chemistry Lectureship: Addressing the “Core Issue” in the Design of Estrogen Receptor Ligands

gan Katzenellenbogen, John A.
Cyhoeddwyd 2011

The Quest for Improving the Management of Breast Cancer by Functional Imaging: The Discovery and Development of 16α-[(18)F]Fluoroestradiol (FES), a PET Radiotracer for the Estrogen...

gan Katzenellenbogen, John A.
Cyhoeddwyd yn Nucl Med Biol (2020)

PET Imaging Agents (FES, FFNP, and FDHT) for Estrogen, Androgen, and Progesterone Receptors to Improve Management of Breast and Prostate Cancers by Functional Imaging

gan Katzenellenbogen, John A.
Cyhoeddwyd yn Cancers (Basel) (2020)

A Dual-Acceptor Time-Resolved Föster Resonance Energy Transfer Assay for Simultaneous Determination of Thyroid Hormone Regulation of Corepressor and Coactivator Binding to the Thyr...

gan Jeyakumar, M., Katzenellenbogen, John A.
Cyhoeddwyd 2008

Designer antiandrogens join the race against drug resistance

gan Josan, Jatinder S, Katzenellenbogen, John A
Cyhoeddwyd 2013

Pyridyl-Cyclopentadiene Re(CO)(2)(+) Complexes as a Compact Core Systems for SPECT Ligand Development

gan Ackroyd, Nathan C., Katzenellenbogen, John A.
Cyhoeddwyd 2010

Improved Chemical Syntheses of 5,6-Dihydro-5-fluorouracil

gan LaFrate, Andrew L., Katzenellenbogen, John A.
Cyhoeddwyd 2007

Dual Mode Fluorophore-Doped Nickel Nitrilotriacetic Acid-Modified Silica Nanoparticles Combine Histidine-Tagged Protein Purification with Site-Specific Fluorophore Labeling

gan Kim, Sung Hoon, Jeyakumar, M., Katzenellenbogen, John A.
Cyhoeddwyd 2007

A New Quinoline Sensitizer-Centered Lanthanide Chelate and Its Use for Protein Labling on Ni-NTA Beads for TR LRET Assays

gan Kim, Sung Hoon, Ge, Pinghua, Katzenellenbogen, John A.
Cyhoeddwyd 2008

Preparation of ortho-Fluorophenols from Non-Aromatic Precursors: Mechanistic Considerations for Adaptation to Fluorine-18 Radiolabeling

gan Yasui, Norio, Mayne, Christopher G., Katzenellenbogen, John A.
Cyhoeddwyd yn Org Lett (2015)

Directed evolution of specific receptor–ligand pairs for use in the creation of gene switches

gan Chockalingam, Karuppiah, Chen, Zhilei, Katzenellenbogen, John A., Zhao, Huimin
Cyhoeddwyd 2005

Blocking Estrogen Signaling After the Hormone: Pyrimidine-Core Inhibitors of Estrogen Receptor-Coactivator Binding

gan Parent, Alexander A., Gunther, Jillian R., Katzenellenbogen, John A.
Cyhoeddwyd 2008

Nonclassical SNAPFL Analog as a Cy5 Resonance Energy Transfer Partner

gan Kim, Sung Hoon, Gunther, Jillian R., Katzenellenbogen, John A.
Cyhoeddwyd 2008

Minireview: Not Picking Pockets: Nuclear Receptor Alternate-Site Modulators (NRAMs)

gan Moore, Terry W., Mayne, Christopher G., Katzenellenbogen, John A.
Cyhoeddwyd 2010

Monitoring a Coordinated Exchange Process in a Four-Component Biological Interaction System: Development of a Time-Resolved Terbium-Based One Donor/Three-Acceptor Multi-Color FRET...

gan Kim, Sung Hoon, Gunther, Jillian R., Katzenellenbogen, John A.
Cyhoeddwyd 2010

Probing the Topological Tolerance of Multimeric Protein Interactions: Evaluation of an Estrogen/Synthetic Ligand for FK506 Binding Protein Conjugate

gan Moore, Terry W., Gunther, Jillian R., Katzenellenbogen, John A.
Cyhoeddwyd 2010

Alternative inhibition of androgen receptor signaling: Peptidomimetic pyrimidines as direct androgen receptor/coactivator disruptors

gan Gunther, Jillian R., Parent, Alexander A., Katzenellenbogen, John A.
Cyhoeddwyd 2009

A New Fluorescence Complementation Biosensor for Detection of Estrogenic Compounds

gan McLachlan, Michael J., Katzenellenbogen, John A., Zhao, Huimin
Cyhoeddwyd 2011

π–π Interaction Energies as Determinants of the Photodimerization of Mono-, Di-, and Triazastilbenes

gan Parent, Alexander A., Ess, Daniel H., Katzenellenbogen, John A.
Cyhoeddwyd 2014

Estrogen Receptors Alpha (ERα) and Beta (ERβ): Subtype-Selective Ligands and Clinical Potential

gan Paterni, Ilaria, Granchi, Carlotta, Katzenellenbogen, John A., Minutolo, Filippo
Cyhoeddwyd 2014