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Selective and potent agonists for estrogen receptor beta derived from molecular refinements of salicylaldoximes

In a continuing effort to improve the subtype selectivity and agonist potency of estrogen receptor β (ERβ) ligands, we have designed and developed a thus far unexplored structural series obtained by molecular refinements of monoaryl-substituted salicylaldoximes (Salaldox B). The most interesting com...

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Detalhes bibliográficos
Main Authors: Bertini, Simone, De Cupertinis, Andrea, Granchi, Carlotta, Bargagli, Barbara, Tuccinardi, Tiziano, Martinelli, Adriano, Macchia, Marco, Gunther, Jillian R., Carlson, Kathryn E., Katzenellenbogen, John A., Minutolo, Filippo
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3088081/
https://ncbi.nlm.nih.gov/pubmed/21481497
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2011.03.030
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