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Anti-infective Activity of 2-Cyano-3-Acrylamide Inhibitors with Improved Drug-Like Properties against Two Intracellular Pathogens

Due to the rise of antibiotic resistance and the small number of effective antiviral drugs, new approaches for treating infectious diseases are urgently needed. Identifying targets for host-based therapies represents an emerging strategy for drug discovery. The ubiquitin-proteasome system is a centr...

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Dettagli Bibliografici
Pubblicato in:Antimicrob Agents Chemother
Autori principali: Passalacqua, Karla D., Charbonneau, Marie-Eve, Donato, Nicholas J., Showalter, Hollis D., Sun, Duxin, Wen, Bo, He, Miao, Sun, Hanshi, O'Riordan, Mary X. D., Wobus, Christiane E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4914689/
https://ncbi.nlm.nih.gov/pubmed/27139470
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.03021-15
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