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Anti-infective Activity of 2-Cyano-3-Acrylamide Inhibitors with Improved Drug-Like Properties against Two Intracellular Pathogens

Due to the rise of antibiotic resistance and the small number of effective antiviral drugs, new approaches for treating infectious diseases are urgently needed. Identifying targets for host-based therapies represents an emerging strategy for drug discovery. The ubiquitin-proteasome system is a centr...

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Publicat a:Antimicrob Agents Chemother
Autors principals: Passalacqua, Karla D., Charbonneau, Marie-Eve, Donato, Nicholas J., Showalter, Hollis D., Sun, Duxin, Wen, Bo, He, Miao, Sun, Hanshi, O'Riordan, Mary X. D., Wobus, Christiane E.
Format: Artigo
Idioma:Inglês
Publicat: American Society for Microbiology 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4914689/
https://ncbi.nlm.nih.gov/pubmed/27139470
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.03021-15
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