Učitavanje...

Rapid Optimization of Mcl-1 Inhibitors using Stapled Peptide Libraries Including Non-Natural Side Chains

Alpha helices form a critical part of the binding interface for many protein-protein interactions, and chemically stabilized synthetic helical peptides can be effective inhibitors of such helix-mediated complexes. In particular, hydrocarbon stapling of peptides to generate constrained helices can im...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Izdano u:ACS Chem Biol
Glavni autori: Araghi, Raheleh Rezaei, Ryan, Jeremy A., Letai, Anthony, Keating, Amy E.
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4874891/
https://ncbi.nlm.nih.gov/pubmed/26854535
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.5b01002
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!