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Rapid Optimization of Mcl-1 Inhibitors using Stapled Peptide Libraries Including Non-Natural Side Chains

Alpha helices form a critical part of the binding interface for many protein-protein interactions, and chemically stabilized synthetic helical peptides can be effective inhibitors of such helix-mediated complexes. In particular, hydrocarbon stapling of peptides to generate constrained helices can im...

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Bibliografiske detaljer
Udgivet i:ACS Chem Biol
Main Authors: Araghi, Raheleh Rezaei, Ryan, Jeremy A., Letai, Anthony, Keating, Amy E.
Format: Artigo
Sprog:Inglês
Udgivet: 2016
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4874891/
https://ncbi.nlm.nih.gov/pubmed/26854535
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.5b01002
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