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Aminoacyl β-naphthylamides as substrates and modulators of AcrB multidrug efflux pump

Efflux pumps of the resistance-nodulation division superfamily, such as AcrB, make a major contribution to multidrug resistance in Gram-negative bacteria. Inhibitors of such pumps would improve the efficacy of antibiotics, and ameliorate the crisis in health care caused by the prevalence of multidru...

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Pubblicato in:Proc Natl Acad Sci U S A
Autori principali: Kinana, Alfred D., Vargiu, Attilio V., May, Thithiwat, Nikaido, Hiroshi
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4747751/
https://ncbi.nlm.nih.gov/pubmed/26787896
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1525143113
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