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Design of composite inhibitors targeting glutamate carboxypeptidase II: the importance of effector functionalities

Inhibitors targeting human glutamate carboxypeptidase II (GCPII) typically consist of a P1’ glutamate-derived binding module, which warrants the high-affinity and specificity, linked to an effector function that is positioned within the entrance funnel of the enzyme. Here we present a comprehensive...

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Bibliografske podrobnosti
izdano v:FEBS J
Main Authors: Novakova, Zora, Cerny, Jiri, Choy, Cindy J., Nedrow, Jessie, Choi, Joeseph K., Lubkowski, Jacek, Berkman, Clifford E., Barinka, Cyril
Format: Artigo
Jezik:Inglês
Izdano: 2015
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC4712110/
https://ncbi.nlm.nih.gov/pubmed/26460595
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/febs.13557
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