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Frequent promoter hypermethylation of PTPRT increases STAT3 activation and sensitivity to STAT3 inhibition in head and neck cancer

STAT3 overactivation is a common event in many cancers, including head and neck squamous cell carcinoma (HNSCC), where STAT3 represents a promising therapeutic target. HNSCC is not characterized by frequent kinase mutations, in contrast to some malignancies where mutational activation of kinases ups...

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Publicat a:Oncogene
Autors principals: Peyser, Noah D., Freilino, Maria, Wang, Lin, Zeng, Yan, Li, Hua, Johnson, Daniel E., Grandis, Jennifer R.
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4651851/
https://ncbi.nlm.nih.gov/pubmed/25982282
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/onc.2015.171
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