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An Aggregation Advisor for Ligand Discovery

Colloidal aggregation of organic molecules is the dominant mechanism for artifactual inhibition of proteins, and controls against it are widely deployed. Notwithstanding an increasingly detailed understanding of this phenomenon, a method to reliably predict aggregation has remained elusive. Correspo...

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Bibliografski detalji
Izdano u:J Med Chem
Glavni autori: Irwin, John J., Duan, Da, Torosyan, Hayarpi, Doak, Allison K., Ziebart, Kristin T., Sterling, Teague, Tumanian, Gurgen, Shoichet, Brian K.
Format: Artigo
Jezik:Inglês
Izdano: 2015
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4646424/
https://ncbi.nlm.nih.gov/pubmed/26295373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01105
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