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An Aggregation Advisor for Ligand Discovery

Colloidal aggregation of organic molecules is the dominant mechanism for artifactual inhibition of proteins, and controls against it are widely deployed. Notwithstanding an increasingly detailed understanding of this phenomenon, a method to reliably predict aggregation has remained elusive. Correspo...

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Publicat a:J Med Chem
Autors principals: Irwin, John J., Duan, Da, Torosyan, Hayarpi, Doak, Allison K., Ziebart, Kristin T., Sterling, Teague, Tumanian, Gurgen, Shoichet, Brian K.
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4646424/
https://ncbi.nlm.nih.gov/pubmed/26295373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01105
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