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An Aggregation Advisor for Ligand Discovery

Colloidal aggregation of organic molecules is the dominant mechanism for artifactual inhibition of proteins, and controls against it are widely deployed. Notwithstanding an increasingly detailed understanding of this phenomenon, a method to reliably predict aggregation has remained elusive. Correspo...

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Detalles Bibliográficos
Publicado en:J Med Chem
Main Authors: Irwin, John J., Duan, Da, Torosyan, Hayarpi, Doak, Allison K., Ziebart, Kristin T., Sterling, Teague, Tumanian, Gurgen, Shoichet, Brian K.
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4646424/
https://ncbi.nlm.nih.gov/pubmed/26295373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01105
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