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Design, Synthesis and Biological evaluation of Multifunctional Ligands Targeting Opioid and Bradykinin 2 Receptors

We report here the design and synthesis of novel multifunctional ligands that act as (μ/δ) opioid agonists and bradykinin 2 receptor antagonists. These multifunctional ligands were designed to interact with the multiple receptors to show an enhanced analgesic effect, with no opioid-induced tolerance...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Main Authors: Deekonda, Srinivas, Rankin, David, Davis, Peg, Lai, Josephine, Porreca, Frank, Hruby, Victor J.
Formato: Artigo
Idioma:Inglês
Publicado: 2015
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4642888/
https://ncbi.nlm.nih.gov/pubmed/26316468
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.08.014
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