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Inhibition of hERG potassium channel by the antiarrhythmic agent mexiletine and its metabolite m-hydroxymexiletine

Mexiletine is a sodium channel blocker, primarily used in the treatment of ventricular arrhythmias. Moreover, recent studies have demonstrated its therapeutic value to treat myotonic syndromes and to relieve neuropathic pain. The present study aims at investigating the direct blockade of hERG potass...

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Опубликовано в: :Pharmacol Res Perspect
Главные авторы: Gualdani, Roberta, Tadini-Buoninsegni, Francesco, Roselli, Mariagrazia, Defrenza, Ivana, Contino, Marialessandra, Colabufo, Nicola Antonio, Lentini, Giovanni
Формат: Artigo
Язык:Inglês
Опубликовано: John Wiley & Sons, Ltd 2015
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4618635/
https://ncbi.nlm.nih.gov/pubmed/26516576
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prp2.160
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