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Radiolabelling and positron emission tomography of PT70, a time-dependent inhibitor of InhA, the Mycobacterium tuberculosis enoyl-ACP reductase

PT70 is a diaryl ether inhibitor of InhA, the enoyl-ACP reductase in the Mycobacterium tuberculosis fatty acid biosynthesis pathway. It has a residence time of 24 min on the target, and also shows antibacterial activity in a mouse model of tuberculosis infection. Due to the interest in studying targ...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Wang, Hui, Liu, Li, Lu, Yang, Pan, Pan, Hooker, Jacob M., Fowler, Joanna S., Tonge, Peter J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4607644/
https://ncbi.nlm.nih.gov/pubmed/26227776
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.07.019
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