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Tight binding enantiomers of pre-clinical drug candidates

MTDIA is a picomolar transition state analogue inhibitor of human methylthioadenosine phosphorylase and a femtomolar inhibitor of E. coli methylthioadenosine nucleosidase. MTDIA has proven to be a non-toxic, orally available pre-clinical drug candidate with remarkable anti-tumour activity against a...

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Bibliografiske detaljer
Udgivet i:Bioorg Med Chem
Main Authors: Evans, Gary B., Cameron, Scott A., Luxenburger, Andreas, Guan, Rong, Suarez, Javier, Thomas, Keisha, Schramm, Vern L., Tyler, Peter C.
Format: Artigo
Sprog:Inglês
Udgivet: 2015
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4567382/
https://ncbi.nlm.nih.gov/pubmed/26260335
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2015.07.059
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