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Tight binding enantiomers of pre-clinical drug candidates

MTDIA is a picomolar transition state analogue inhibitor of human methylthioadenosine phosphorylase and a femtomolar inhibitor of E. coli methylthioadenosine nucleosidase. MTDIA has proven to be a non-toxic, orally available pre-clinical drug candidate with remarkable anti-tumour activity against a...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Bioorg Med Chem
Päätekijät: Evans, Gary B., Cameron, Scott A., Luxenburger, Andreas, Guan, Rong, Suarez, Javier, Thomas, Keisha, Schramm, Vern L., Tyler, Peter C.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2015
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC4567382/
https://ncbi.nlm.nih.gov/pubmed/26260335
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2015.07.059
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