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High-throughput screening by Nuclear Magnetic Resonance (HTS by NMR) for the identification of PPIs antagonists

In recent years the ever so complex field of drug discovery has embraced novel design strategies based on biophysical fragment screening (fragment-based drug design; FBDD) using nuclear magnetic resonance spectroscopy (NMR) and/or structure-guided approaches, most often using X-ray crystallography a...

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Publicat a:Curr Top Med Chem
Autors principals: Wu, Bainan, Barile, Elisa, De, Surya K., Wei, Jun, Purves, Angela, Pellecchia, Maurizio
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4545611/
https://ncbi.nlm.nih.gov/pubmed/25986689
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