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A β-Fluoroamine Inhibitor of Purine Nucleoside Phosphorylase

The potent immucillin purine nucleoside phosphorylase (PNP) inhibitors F-DADMe-ImmH [(3S,4S)−3], and [(3R,4R)−3] are synthesized in seven steps. Cycloaddition to a fluoroalkene and an enzymic resolution are the key features of the construction of the fluoropyrrolidines 11, from which the immucillins...

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Détails bibliographiques
Publié dans:J Med Chem
Auteurs principaux: Mason, Jennifer M., Murkin, Andrew S., Li, Lei, Schramm, Vern L., Gainsford, Graeme J., Skelton, Brian W.
Format: Artigo
Langue:Inglês
Publié: 2008
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4508846/
https://ncbi.nlm.nih.gov/pubmed/18800772
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm800792b
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