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Diphenyl Purine Derivatives as Peripherally Selective Cannabinoid Receptor 1 Antagonists

Cannabinoid receptor 1 (CB1) antagonists are potentially useful for the treatment of several diseases. However, clinical development of several CB1 antagonists was halted due to central nervous system (CNS)-related side effects including depression and suicidal ideation in some users. Recently, stud...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Fulp, Alan, Bortoff, Katherine, Zhang, Yanan, Seltzman, Herbert, Mathews, James, Snyder, Rodney, Fennell, Tim, Maitra, Rangan
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4492447/
https://ncbi.nlm.nih.gov/pubmed/23098108
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301181r
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