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Structure-Guided, Single-Point Modifications in the Phosphinic Dipeptide Structure Yield Highly Potent and Selective Inhibitors of Neutral Aminopeptidases

[Image: see text] Seven crystal structures of alanyl aminopeptidase from Neisseria meningitides (the etiological agent of meningitis, NmAPN) complexed with organophosphorus compounds were resolved to determine the optimal inhibitor–enzyme interactions. The enantiomeric phosphonic acid analogs of Leu...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Vassiliou, Stamatia, Węglarz-Tomczak, Ewelina, Berlicki, Łukasz, Pawełczak, Małgorzata, Nocek, Bogusław, Mulligan, Rory, Joachimiak, Andrzej, Mucha, Artur
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2014
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4331105/
https://ncbi.nlm.nih.gov/pubmed/25192493
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm501071f
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