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PQ-69, a novel and selective adenosine A(1) receptor antagonist with inverse agonist activity

Potent and selective adenosine A(1) receptor (A(1)AR) antagonists with favourable pharmacokinetic properties used as novel diuretics and antihypertensives are desirable. Thus, we designed and synthesized a series of novel 4-alkylamino substitution-2-arylpyrazolo[4,3-c]quinolin-3-one derivatives. The...

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Dades bibliogràfiques
Publicat a:Purinergic Signal
Autors principals: Lu, Min, Wang, Bo, Zhang, Cheng, Zhuang, Xiaomei, Yuan, Mei, Wang, Haoshan, Li, Weizhang, Su, Ruibin, Li, Jin
Format: Artigo
Idioma:Inglês
Publicat: Springer Netherlands 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4272367/
https://ncbi.nlm.nih.gov/pubmed/25248972
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11302-014-9424-5
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