Carregant...

Effect of chirality and lipophilicity in the functional activity of evodiamine and its analogues at TRPV1 channels

BACKGROUND AND PURPOSE: Evodiamine, a racemic quinazolinocarboline alkaloid isolated from the traditional Chinese medicine Evodiae fructus, has been reported to act as an agonist of the transient receptor potential vanilloid type-1 (TRPV1) cation channel both in vitro and in vivo. Evodiamine is stru...

Descripció completa

Guardat en:
Dades bibliogràfiques
Autors principals: De Petrocellis, Luciano, Schiano Moriello, Aniello, Fontana, Gabriele, Sacchetti, Alessandro, Passarella, Daniele, Appendino, Giovanni, Di Marzo, Vincenzo
Format: Artigo
Idioma:Inglês
Publicat: Blackwell Publishing Ltd 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4009003/
https://ncbi.nlm.nih.gov/pubmed/23902373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.12320
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!