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Conformation-selective inhibitors reveal differences in the activation and phosphate-binding loops of the tyrosine kinases Abl and Src

Over the last decade, an increasingly diverse array of potent and selective inhibitors that target the ATP-binding sites of protein kinases have been developed. Many of these inhibitors, like the clinically approved drug imatinib (Gleevec), stabilize a specific catalytically inactive ATP-binding sit...

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Détails bibliographiques
Auteurs principaux: Hari, Sanjay B., Perera, B. Gayani K., Ranjitkar, Pratistha, Seeliger, Markus A., Maly, Dustin J.
Format: Artigo
Langue:Inglês
Publié: 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3880807/
https://ncbi.nlm.nih.gov/pubmed/24106839
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb400663k
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