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Bivalent inhibitors of the tyrosine kinases ABL and SRC: Determinants of potency and selectivity

We recently reported a chemical genetic method for generating bivalent inhibitors of protein kinases. This method relies on the use of the DNA repair enzyme O(6)-alkylguanine-DNA alkyltransferase (AGT) to display an ATP-competitive inhibitor and a ligand that targets a secondary binding domain. With...

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Detalhes bibliográficos
Main Authors: Hill, Zachary B., Perera, B. Gayani K., Maly, Dustin J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3268058/
https://ncbi.nlm.nih.gov/pubmed/21060940
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c0mb00108b
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