Yüklüyor......

Bivalent inhibitors of the tyrosine kinases ABL and SRC: Determinants of potency and selectivity

We recently reported a chemical genetic method for generating bivalent inhibitors of protein kinases. This method relies on the use of the DNA repair enzyme O(6)-alkylguanine-DNA alkyltransferase (AGT) to display an ATP-competitive inhibitor and a ligand that targets a secondary binding domain. With...

Ful tanımlama

Kaydedildi:
Detaylı Bibliyografya
Asıl Yazarlar: Hill, Zachary B., Perera, B. Gayani K., Maly, Dustin J.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2010
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC3268058/
https://ncbi.nlm.nih.gov/pubmed/21060940
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c0mb00108b
Etiketler: Etiketle
Etiket eklenmemiş, İlk siz ekleyin!