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Substituted Tetrahydroisoquinolines as Selective Antagonists for the Orexin 1 Receptor

Increasing evidence implicates the orexin 1 (OX(1)) receptor in reward processes, suggesting OX(1) antagonism could be therapeutic in drug addiction. In a program to develop an OX(1) selective antagonist, we designed and synthesized a series of substituted tetrahydroisoquinolines and determined thei...

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Detalhes bibliográficos
Main Authors: Perrey, David A., German, Nadezhda A., Gilmour, Brian P., Li, Jun-Xu, Harris, Danni L., Thomas, Brian F., Zhang, Yanan
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3849818/
https://ncbi.nlm.nih.gov/pubmed/23941044
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm400720h
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