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The cyclin-dependent kinase inhibitor dinaciclib interacts with the acetyl-lysine recognition site of bromodomains

Bromodomain-containing proteins are considered atypical kinases, but their potential to interact with kinase inhibitors is unknown. Dinaciclib is a potent inhibitor of cyclin-dependent kinases (CDKs) which recently advanced to Phase III clinical trials for the treatment of leukemia. We determined th...

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Autors principals: Martin, Mathew P., Olesen, Sanne H., Georg, Gunda I., Schönbrunn, Ernst
Format: Artigo
Idioma:Inglês
Publicat: 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3846258/
https://ncbi.nlm.nih.gov/pubmed/24007471
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb4003283
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