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Structural Basis of Wee Kinases Functionality and Inactivation by Diverse Small Molecule Inhibitors

Members of the Wee family of kinases negatively regulate the cell cycle via phosphorylation of CDK1 and are considered potential drug targets. Herein, we investigated the structure–function relationship of human Wee1, Wee2, and Myt1 (PKMYT1). Purified recombinant full-length proteins and kinase doma...

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Détails bibliographiques
Publié dans:J Med Chem
Auteurs principaux: Zhu, Jin-Yi, Cuellar, Rebecca A., Berndt, Norbert, Lee, Hee Eun, Olesen, Sanne H., Martin, Mathew P., Jensen, Jeffrey T., Georg, Gunda I., Schönbrunn, Ernst
Format: Artigo
Langue:Inglês
Publié: 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6200136/
https://ncbi.nlm.nih.gov/pubmed/28792760
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.7b00996
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