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Piperine activates human pregnane X receptor to induce the expression of cytochrome P450 3A4 and multidrug resistance protein 1

Activation of the pregnane X receptor (PXR) and subsequently its target genes, including those encoding drug transporters and metabolizing enzymes, while playing substantial roles in xenobiotics detoxification, might cause undesired drug-drug interactions. Recently, an increased awareness has been g...

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Autores principales: Wang, Yue-Ming, Lin, Wenwei, Chai, Sergio C., Wu, Jing, Ong, Su Sien, Schuetz, Erin G., Chen, Taosheng
Formato: Artigo
Lenguaje:Inglês
Publicado: 2013
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3775940/
https://ncbi.nlm.nih.gov/pubmed/23707768
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.taap.2013.05.014
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