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Identification and Characterization of Phosphorylation Sites within the Pregnane X Receptor Protein

Pregnane X receptor (PXR) is a xenobiotic sensor regulating the expression of genes involved in xenobiotic detoxification and elimination. Phosphorylation plays an important role in modulating PXR activity and several phosphorylation sites have been predicted and characterized in in vitro experiment...

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Autors principals: Elias, Ayesha, High, Anthony A., Mishra, Ashutosh, Ong, Su Sien, Wu, Jing, Peng, Junmin, Chen, Taosheng
Format: Artigo
Idioma:Inglês
Publicat: 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3947193/
https://ncbi.nlm.nih.gov/pubmed/24184507
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2013.10.015
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