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Stability of the human pregnane X receptor is regulated by E3 ligase UBR5 and serine/threonine kinase DYRK2

The human pregnane X receptor (hPXR), a major chemical toxin sensor, is a ligand-induced transcription factor activated by various xenobiotics and toxins, resulting in the transcriptional upregulation of detoxifying enzymes. To date, little is known about the upstream regulation of hPXR. Using mass...

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Autors principals: Ong, Su Sien, Goktug, Asli N., Elias, Ayesha, Wu, Jing, Saunders, Darren, Chen, Taosheng
Format: Artigo
Idioma:Inglês
Publicat: 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3959618/
https://ncbi.nlm.nih.gov/pubmed/24438055
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20130558
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