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Contribution of Abcc4-Mediated Gastric Transport to the Absorption and Efficacy of Dasatinib

PURPOSE: Several oral multikinase inhibitors are known to interact in vitro with the human ATP-binding cassette transporter ABCC4 (MRP4), but the in vivo relevance of this interaction remains poorly understood. We hypothesized that host ABCC4 activity may influence the pharmacokinetic profile of das...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Furmanski, Brian D., Hu, Shuiying, Fujita, Ken-ichi, Li, Lie, Gibson, Alice A., Janke, Laura J., Williams, Richard T., Schuetz, John D., Sparreboom, Alex, Baker, Sharyn D.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2013
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3752901/
https://ncbi.nlm.nih.gov/pubmed/23794731
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-13-0980
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