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Design, Synthesis and Biological Activity of Multifunctional α,β- Unsaturated Carbonyl Scaffolds for Alzheimer’s Disease

A series of compounds containing an α,β-unsaturated carbonyl moiety, such as chalcones and coumarins were designed, synthesized and tested in a variety of assays to assess their potential as anti-Alzheimers’ disease (AD) agents. The investigations included the inhibition of cholinesterases (AChE, Bu...

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Autors principals: Bag, Seema, Ghosh, Sanjukta, Tulsan, Rekha, Sood, Abha, Zhou, Weihong, Schifone, Christine, Foster, Michelle, LeVine, Harry, Török, Béla, Török, Marianna
Format: Artigo
Idioma:Inglês
Publicat: 2013
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3676911/
https://ncbi.nlm.nih.gov/pubmed/23540646
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.02.103
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