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Reversible targeting of noncatalytic cysteines with chemically tuned electrophiles

Targeting noncatalytic cysteine residues with irreversible acrylamide-based inhibitors is a powerful approach for enhancing pharmacological potency and selectivity. Nevertheless, concerns about off-target modification motivate the development of reversible cysteine-targeting strategies. Here we show...

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Detalhes bibliográficos
Main Authors: Serafimova, Iana M., Pufall, Miles A., Krishnan, Shyam, Duda, Katarzyna, Cohen, Michael S., Maglathlin, Rebecca L., McFarland, Jesse M., Miller, Rand M., Frödin, Morten, Taunton, Jack
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3657615/
https://ncbi.nlm.nih.gov/pubmed/22466421
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.925
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