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Interaction of human cytochrome P4503A4 with ritonavir analogs

Ritonavir is a HIV protease inhibitor that also potently inactivates cytochrome P450 3A4 (CYP3A4), a major human drug-metabolizing enzyme. To better understand the mechanism of ligand binding and to find strategies for improvement of the inhibitory potency of ritonavir, currently administered to enh...

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Bibliografski detalji
Glavni autori: Sevrioukova, Irina F., Poulos, Thomas L.
Format: Artigo
Jezik:Inglês
Izdano: 2012
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3606017/
https://ncbi.nlm.nih.gov/pubmed/22410611
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.abb.2012.02.018
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