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Structure and mechanism of the complex between cytochrome P4503A4 and ritonavir

Ritonavir is a HIV protease inhibitor routinely prescribed to HIV patients that also potently inactivates cytochrome P4503A4 (CYP3A4), the major human drug-metabolizing enzyme. By inhibiting CYP3A4, ritonavir increases plasma concentrations of other anti-HIV drugs oxidized by CYP3A4 thereby improvin...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Sevrioukova, Irina F., Poulos, Thomas L.
Format: Artigo
Sprache:Inglês
Veröffentlicht: National Academy of Sciences 2010
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2973003/
https://ncbi.nlm.nih.gov/pubmed/20937904
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1010693107
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