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Discovery of Highly Potent and Selective α4β2-Nicotinic Acetylcholine Receptor (nAChR) Partial Agonists Containing an Isoxazolylpyridine Ether Scaffold that Demonstrate Antidepressant-like Activity. Part II

In our continued efforts to develop α4β2-nicotinic acetylcholine receptor (nAChR) partial agonists as novel antidepressants having a unique mechanism of action, structure activity relationship (SAR) exploration of certain isoxazolylpyridine ethers is presented. In particular, modifications to both t...

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Библиографические подробности
Главные авторы: Yu, Li-Fang, Eaton, J. Brek, Fedolak, Allison, Zhang, Han-Kun, Hanania, Taleen, Brunner, Dani, Lukas, Ronald J., Kozikowski, Alan P.
Формат: Artigo
Язык:Inglês
Опубликовано: 2012
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3532055/
https://ncbi.nlm.nih.gov/pubmed/23092294
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301177j
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