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Catalytic activities of a cocaine hydrolase engineered from human butyrylcholinesterase against (+)- and (−)-cocaine

It can be argued that an ideal anti-cocaine medication would be one that accelerates cocaine metabolism producing biologically inactive metabolites via a route similar to the primary cocaine-metabolizing pathway, i.e. hydrolysis catalyzed by butyrylcholinesterase (BChE) in plasma. However, wild-type...

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Autori principali: Xue, Liu, Hou, Shurong, Yang, Wenchao, Fang, Lei, Zheng, Fang, Zhan, Chang-Guo
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3527670/
https://ncbi.nlm.nih.gov/pubmed/22917637
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.cbi.2012.08.003
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