Carregant...

The importance of the trans-enamine intermediate as a β-lactamase inhibition strategy probed in inhibitor-resistant SHV β-lactamase variants

The ability of bacteria expressing inhibitor resistant (IR) β-lactamases is stimulating the development of novel inhibitors. SA2-13 was previously designed to enhance the stabilization of the deacylation refractory, trans-enamine inhibitory intermediate. To test whether this mode of inhibition can o...

Descripció completa

Guardat en:
Dades bibliogràfiques
Autors principals: Ke, Wei, Rodkey, Elizabeth A., Sampson, Jared M., Skalweit, Marion J., Sheri, Anjaneyulu, Pagadala, Sundar Ram Reddy, Nottingham, Michael D., Buynak, John D., Bonomo, Robert A., van den Akker, Focco
Format: Artigo
Idioma:Inglês
Publicat: 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3523351/
https://ncbi.nlm.nih.gov/pubmed/22438274
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201200006
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!