טוען...

Steric Hindrance Mutagenesis in the Conserved Extracellular Vestibule Impedes Allosteric Binding of Antidepressants to the Serotonin Transporter

The serotonin transporter (SERT) controls synaptic serotonin levels and is the primary target for antidepressants, including selective serotonin reuptake inhibitors (e.g. (S)-citalopram) and tricyclic antidepressants (e.g. clomipramine). In addition to a high affinity binding site, SERT possesses a...

תיאור מלא

שמור ב:
מידע ביבליוגרפי
Main Authors: Plenge, Per, Shi, Lei, Beuming, Thijs, Te, Jerez, Newman, Amy Hauck, Weinstein, Harel, Gether, Ulrik, Loland, Claus J.
פורמט: Artigo
שפה:Inglês
יצא לאור: American Society for Biochemistry and Molecular Biology 2012
נושאים:
גישה מקוונת:https://ncbi.nlm.nih.gov/pmc/articles/PMC3501018/
https://ncbi.nlm.nih.gov/pubmed/23007398
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M112.371765
תגים: הוספת תג
אין תגיות, היה/י הראשונ/ה לתייג את הרשומה!