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High-affinity and selective dopamine D(3) receptor full agonists

We have designed, synthesized and evaluated a series of new compounds with the goal to identify potent and selective D(3) ligands. The two most potent and selective new D(3) ligands are compounds 38 and 52, which bind to the D(3) receptors with a K(i) value of <1 nM and display a selectivity of 4...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Chen, Jianyong, Levant, Beth, Wang, Shaomeng
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2012
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3461280/
https://ncbi.nlm.nih.gov/pubmed/22871578
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2012.07.003
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