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Design, Synthesis and Evaluation of Potent and Selective Ligands for the Dopamine 3 (D(3)) Receptor with a Novel in vivo Behavioral Profile

A series of compounds structurally related to pramipexole were designed, synthesized and evaluated as ligands for the dopamine 3 (D(3)) receptor. Compound 12 has a K(i) value of 0.41 nM to D(3) and a selectivity of >30,000- and 800-fold over the D(1)-like and D(2) receptors, respectively. Our in...

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Detalhes bibliográficos
Main Authors: Chen, Jianyong, Collins, Gregory T., Zhang, Jian, Yang, Chao-Yie, Levant, Beth, Woods, James, Wang, Shaomeng
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2662387/
https://ncbi.nlm.nih.gov/pubmed/18785726
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm800471h
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