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Light-regulation of protein dimerization and kinase activity in living cells using photocaged rapamycin and engineered FKBP

[Image: see text] We developed a new system for light-induced protein dimerization in living cells using a novel photocaged analog of rapamycin (pRap) together with an engineered rapamycin binding domain (iFKBP). Using focal adhesion kinase as a target, we demonstrated successful light-mediated regu...

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Detalhes bibliográficos
Main Authors: Karginov, Andrei V., Zou, Yan, Shirvanyants, David, Kota, Pradeep, Dokholyan, Nikolay V., Young, Douglas D., Hahn, Klaus M., Deiters, Alexander
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3133816/
https://ncbi.nlm.nih.gov/pubmed/21162531
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja109630v
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