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Interactions between the Etoposide Derivative F14512 and Human Type II Topoisomerases: Implications for the C4 Spermine Moiety in Promoting Enzyme-mediated DNA Cleavage

F14512 is a novel etoposide derivative that contains a spermine in place of the C4 glycosidic moiety. The drug was designed to exploit the polyamine transport system that is upregulated in some cancers. However, a preliminary study suggests that it is also a more efficacious topoisomerase II poison...

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Bibliografiset tiedot
Päätekijät: Gentry, Amanda C., Pitts, Steven L., Jablonsky, Michael J., Bailly, Christian, Graves, David E., Osheroff, Neil
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2011
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC3086367/
https://ncbi.nlm.nih.gov/pubmed/21413765
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi200094z
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