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Triterpene Derivatives that Inhibit Human Immunodeficiency Virus Type 1 Replication

Triterpene derivatives were analyzed for anti-HIV-1 activity and for cellular toxicity. Betulinic aldehyde, betulinic nitrile, and morolic acid derivatives were identified to have anti-HIV-1 activity. These derivatives inhibit a late step in virus replication, likely virus maturation.

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Dades bibliogràfiques
Autors principals: Dorr, Casey R., Yemets, Sergiy, Kolomitsyna, Oksana, Krasutsky, Pavel, Mansky, Louis M.
Format: Artigo
Idioma:Inglês
Publicat: 2011
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3053071/
https://ncbi.nlm.nih.gov/pubmed/21084190
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2010.10.078
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